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Product Name | AS-2717638 |
Description | An LPA5 antagonist (IC50 = 0.038 µM); selective for LPA5 over LPA1, LPA2, and LPA3 (IC50s = >10 µM for all) but also binds to adenosine A1 and μ-opioid receptors at 10 µM; induces analgesia in a rat model of allodynia induced by LPA or GGPP; inhibits allodynia induced by PGE2, PGF2α, or AMPA in rats at 10 and 30 mg/kg; increases the paw withdrawal threshold and latency in the von Frey hair and plantar tests, respectively, in rats at 10 mg/kg |
Size | 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | AS2717638 LPA-5 1 2 3 geranyl PGE-2 PGF-2α vonFrey |
Gene, Accession, CAS # | CAS: 2148339-28-8 |
Catalog # | 37787-5 |
Price | $336.00 |
Order / More Info | AS-2717638 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |