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Product Name | CPI-637 |
Description | An inhibitor of CBP/EP300 bromodomains (IC50s = 30 and 51 nM in a TR-FRET assay); selective for CBP and EP300 over the BET family of bromodomains (IC50s = >10 µM); is active at bromodomain BRD9 (IC50 = 0.73 µM); inhibits CBP (IC50 = 0.3 µM in a BRET assay) and inhibits MYC expression (EC50 = 0.6 µM) in AMO-1 cells |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | CPI637 fluorescence resonance energy transfer cAMP EP-300 TRFRET BRD-9 AMO1 |
Gene, Accession, CAS # | CAS: 1884712-47-3 |
Catalog # | 23500-1 |
Price | $32.00 |
Order / More Info | CPI-637 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |