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Product Name | CP 80,633 |
Description | A selective inhibitor of PDE4 (IC50 = 1.27 µM for PDE4 versus >100 µM for PDE1, PDE2, PDE3, and PDE5); inhibits eosinophil superoxide production (IC50 induced TNFα release from monocytes ,(IC50 = 0.22 µM); significantly reduces antigen-induced airway inflammation in atopic guinea pigs, monkeys, and mice |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | phosphodiesterases PDE cAMP cGMP asthma neurological diseases inhibitors inhibits inhibition PDE4 PDE1 PDE2 PDE3 PDE5 inflammation CP-80,633 CP-806333 CP80633 Pyrimidinones Pyrimidones |
Gene, Accession, CAS # | CAS: 135637-46-6 |
Catalog # | 13183-10 |
Price | $357.00 |
Order / More Info | CP 80,633 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |