Edit |   |
---|---|
Product Name | Regorafenib N-oxide |
Description | An active metabolite of regorafenib; formed from regorafenib by CYP3A4; inhibits VEGFR2, Tie2, c-Kit, and B-RAF in vitro; inhibits tumor growth in HT-29 and MDA-MB-231 mouse xenograft models at 1 mg/kg |
Size | 25 mg |
Concentration | n/a |
Applications | n/a |
Other Names | Noxide CYP450 CYP 3A4 VEGFR 2 Tie 2 cKit BRAF HT29 MDAMB231 Metabolite M2 |
Gene, Accession, CAS # | CAS: 835621-11-9 |
Catalog # | 35101-25 |
Price | $456 |
Order / More Info | Regorafenib N-oxide from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |