ARV-771 from CAYMAN CHEMICAL COMPANY
Search, find, compare suppliers for ARV-771 products.
| Edit | |
|---|---|
| Product Name | ARV-771 |
| Description | A PROTAC that drives BET family protein degradation; induces degradation of BRD2, BRD3, and BRD4 in 22Rv1 CRPC cells (DC50s = <5 nM for all); inhibits proliferation of and increases PARP cleavage in 22Rv1 cells in a concentration-dependent manner; reduces full-length androgen receptor protein levels and prevents R1881-induced increases in ERG in VCaP cells; induces tumor regression in a 22Rv1 mouse xenograft model at 30 mg/kg per day, s.c. |
| Size | 1 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | ARV771 BRD-2 BRD-3 BRD-4 E-3 R-1881 |
| Gene, Accession, CAS # | CAS: 1949837-12-0 |
| Catalog # | 21299-1 |
| Price | $57.00 |
| Order / More Info | ARV-771 from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640
Customer Service: custserv@caymanchem.com
Technical Support: techserv@caymanchem.com
Sales: sales@caymanchem.com
http://www.caymanchem.com
Profile of CAYMAN CHEMICAL COMPANY