MSC2530818 from CAYMAN CHEMICAL COMPANY
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| Product Name | MSC2530818 |
| Description | A Cdk8 inhibitor (IC50 = 2.6 nM); selective for Cdk8 over a panel of 264 kinases at 1 µM but does inhibit GSK3α (IC50 = 691 nM); inhibits STAT1 phosphorylation in SW620 colorectal cancer cells (IC50 = 8 nM); inhibits Wnt-dependent transcription in LS 174T, COLO 205, and PA-1 cancer cells (IC50s = 32, 9, and 52 nM, respectively, in luciferase reporter assays); reduces tumor growth in a SW620 mouse xenograft model at 50 and 100 mg/kg |
| Size | 25 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | MSC 2530818 bio available Cdk 8 SW 620 174 T PA1 STAT 1 LS174T COLO205 GSK 3 α |
| Gene, Accession, CAS # | CAS: 1883423-59-3 |
| Catalog # | 29669-25 |
| Price | $717.00 |
| Order / More Info | MSC2530818 from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640
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http://www.caymanchem.com
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