O-Desmethyl Gefitinib from CAYMAN CHEMICAL COMPANY

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Product NameO-Desmethyl Gefitinib
DescriptionA major active metabolite of gefitinib in human plasma; inhibits EGFR in subcellular assays similarly to gefitinib (IC50s = 36 and 22 nM, respectively); less active than gefitinib in whole cell assays (IC50s = 760 and 49 nM, respectively); does not reduce tumor growth as well as gefitinib in a LoVo tumor mouse xenograft model,
Size5 mg
Concentrationn/a
Applicationsn/a
Other NamesCYP450 2D6 endothelial growth factor receptor M523595 M-523595
Gene, Accession, CAS #CAS: 847949-49-9
Catalog #22365-5
Price$160.00
Order / More InfoO-Desmethyl Gefitinib from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640

Customer Service: custserv@caymanchem.com
Technical Support: techserv@caymanchem.com
Sales: sales@caymanchem.com

http://www.caymanchem.com

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