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Product Name | EPZ6438 |
Description | An orally bioavailable, selective inhibitor of EZH2 (Ki = 2.5 nM); blocks H3K27 trimethylation in both wild-type and mutant lymphoma cells (IC50s range from 2-90 nM); induces apoptosis and differentiation specifically in SMARCB1-deleted malignant rhabdoid tumor cells and promotes their regression in xenograft-bearing mice |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | Tazemetostat |
Gene, Accession, CAS # | CAS: 1403254-99-8 |
Catalog # | 16174-1 |
Price | $44.00 |
Order / More Info | EPZ6438 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |