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Product Name | Q94 (hydrochloride hydrate) |
Description | A Gαq signaling-biased PAR1 antagonist (IC50 = 916 nM); inhibits thrombin- or a PAR1-activating peptide-induced increases in intracellular calcium mobilization in HMEC-1 cells at 1 and 10 µM; decreases albuminuria in a doxorubicin-induced mouse model of nephropathy at 5 mg/kg per day |
Size | 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 537009-12-4 1052076-77-3 HCl Q-94 Gα PAR HMEC1 |
Gene, Accession, CAS # | n/a |
Catalog # | 32857-5 |
Price | $145 |
Order / More Info | Q94 (hydrochloride hydrate) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |