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Product Name | TP-238 (hydrochloride) |
Description | A chemical probe for CECR2 and BPTF bromodomains; has on-target biochemical activity with CECR2 at 10-30 nM and with BPTF at 100-350 nM; selective for the CECR2 and BPTF bromodomains over BRD9 (IC50 = 1.4 µM), as well as over a panel of 338 kinases at 1 µM; binds to CECR2 and BPTF in ITC (KDs =10 and 120 nM, respectively) and AlphaScreen® assays (IC50s - 30 and 350 nM, respectively) |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | TP238 CECR-2 BRD9 |
Gene, Accession, CAS # | CAS: 2415263-05-5 |
Catalog # | 27254-10 |
Price | $508.00 |
Order / More Info | TP-238 (hydrochloride) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |