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Product Name | VU0152100 |
Description | A positive allosteric modulator of M4 muscarinic acetylcholine receptors; potentiates ACh-induced calcium mobilization in CHO-K1 cells expressing the rat M4 receptor (EC50 = 380 nM); selective for M4 over M1, M2, M3 and M5 receptors, as well as a panel of 68 additional GPCRs, ion channels, transporters, and enzymes but does bind to the benzodiazepine binding site of the GABAA receptor at 10 µM; reduces cocaine-induced increases in locomotor activity and cocaine self-administration in mice at 1 mg/kg |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 1613733-57-5 VU 0152100 GABA A ML 108 ML108 |
Gene, Accession, CAS # | CAS: 409351-28-6 |
Catalog # | 32968-10 |
Price | $158.00 |
Order / More Info | VU0152100 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |