Lys-(Des-Arg9, Leu8)-Bradykinin (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY

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Product NameLys-(Des-Arg9, Leu8)-Bradykinin (trifluoroacetate salt)
DescriptionA bradykinin B1 receptor antagonist (Ki = 0.43 nM for the rabbit aorta receptor); selective for the bradykinin B1 over the B2 receptor (Ki = >10 µM for the rabbit ileum receptor); inhibits contractions induced by Des-Arg9-bradykinin in isolated rabbit aortic rings (pA2 = 8.54); intraperitoneal administration reduces increases in paw edema in a rat model of PGPS-induced arthritis at 5 mg/kg per day for three days
Size25 mg
Concentrationn/a
Applicationsn/a
Other Names[Des-Arg10,Leu9]-Kallidin|[Des-Arg10,Leu9]-KD|Lys[Leu8]Des-Arg9-BK|Lys[Leu8]Des-Arg9-Bradykinin
Gene, Accession, CAS #n/a
Catalog #35462-25
Price$311.00
Order / More InfoLys-(Des-Arg9, Leu8)-Bradykinin (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640

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