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Product Name | TP-3654 |
Description | A Pim kinase inhibitor (Kis = 5, 239, and 42 nM for Pim-1, Pim-2, and Pim-3, respectively); inhibits 19 additional kinases, including PI3Kα, PI3Kγ, and PI3Kδ, with IC50 values 50 = 67 nM), as well as in UM-UC-3 cells; reduces tumor growth in UM-UC-3 bladder carcinoma and PC3 prostate adenocarcinoma mouse xenograft models at 200 mg/kg |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | TP3654 Pim1 Pim2 Pim3 α PI3K-γ δ HEK-293 UMUC UMUC3 PC-3 |
Gene, Accession, CAS # | CAS: 1361951-15-6 |
Catalog # | 29571-10 |
Price | $107.00 |
Order / More Info | TP-3654 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |