TD-4208 from CAYMAN CHEMICAL COMPANY
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| Product Name | TD-4208 |
| Description | An antagonist of muscarinic acetylcholine receptors (Kis = 0.42, 0.3, 0.18, and 0.55 nM for M1, M2, M3, and M4 receptors, respectively, in CHO-K1 cell membranes with the human receptors); selective for these receptors over M5 muscarinic receptors (Ki = 6.31 nM in CHO-K1 cell membranes with the human receptor); inhibits AChE-induced calcium mobilization in CHO-K1 cells expressing M2 and M3 muscarinic receptors; decreases AChE-induced contractions in isolated rat trachea in a concentration-dependent manner; decreases AChE-induced bronchoconstriction and reduces pilocarpine-induced salivation, a surrogate test for noisy breathing, in rats (ID50s = 45 and 1,164 µg/ml, respectively); decreases AChE-induced bronchoconstriction in dogs at 10 and 30 µg/kg intranasally |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | Revefenacin |
| Gene, Accession, CAS # | CAS: 864750-70-9 |
| Catalog # | 36549-10 |
| Price | $36.00 |
| Order / More Info | TD-4208 from CAYMAN CHEMICAL COMPANY |
| Product Specific References | n/a |
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640
Customer Service: custserv@caymanchem.com
Technical Support: techserv@caymanchem.com
Sales: sales@caymanchem.com
http://www.caymanchem.com
Profile of CAYMAN CHEMICAL COMPANY