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Product Name | M40 (trifluoroacetate salt) |
Description | A GAL1 and GAL2 receptor modulator (Kis = 2.4 and 4.07 nM, respectively); selective for GAL1 and GAL2 over GAL3 (Ki = 288 nM); induces inositol phosphate accumulation in CHO cells expressing the human GAL2 receptor (EC50 = 16.2 nM); inhibits forskolin-induced cAMP accumulation in RIN-m5F cells at 10 or 100 nM; reverses galanin-induced inhibition of scopolamine-induced hippocampal ACh release in conscious rats at 9.36 nmol/animal, i.c.v.; reduces galanin-induced increases in food intake in rats; improves cardiac function and decreases cardiac fibrosis in a rat model of heart failure induced by sustained coronary artery ligation at 30 nmol/kg; increases the intromission frequency and ejaculation latency in sexually sluggish male mice at 20 µg/animal |
Size | 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | Galanin-(1-12)-Pro3-(Ala-Leu)2-Ala amide |
Gene, Accession, CAS # | n/a |
Catalog # | 39726-5 |
Price | $956.00 |
Order / More Info | M40 (trifluoroacetate salt) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |