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Product Name | LP-935509 |
Description | An AAK1 and BIKe inhibitor (IC50s = 3.3 and 14 nM, respectively); selective for AAK1 and BIKe over μ- and κ-opioid, as well as α2A- and α2C-adrenergic, receptors (IC50s = >30 µM for all), α1 and α2 subunit-containing GABAA receptors (IC50s = 12 µM for both), and GAK (IC50 = 0.32 µM); reduces phosphorylation of AP2M1 in SH-SY5Y cells at 1 µM; reduces the number of formalin-induced flinches in mice at 10, 30, and 60 mg/kg |
Size | 10 mg |
Concentration | n/a |
Applications | n/a |
Other Names | LP935509 AAK-1 BMP-2 AP2-M1 SHSY5Y |
Gene, Accession, CAS # | CAS: 1454555-29-3 |
Catalog # | 37283-10 |
Price | $299.00 |
Order / More Info | LP-935509 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |