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Product Name | BMS 986122 |
Description | A positive allosteric modulator of μ-opioid receptors (EC50 = 3 µM for endomorphin 1-stimulated β-arrestin recruitment in U2OS-OPRM1 cells expressing human μ-opioid receptors); potentiates endomorphin 1-induced inhibition of forskolin-stimulated adenylyl cyclase activity in CHO cells expressing human μ-opioid receptors (EC50 = 8.9 µM); enhances DAMGO-stimulated [35S]GTPγ binding in C6μ glioma cell membranes and mouse brain membranes |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | BMS986122 U2OSOPRM1 U2O-S OPRM-1 Chinese hamster ovary C-6μ 6 |
Gene, Accession, CAS # | CAS: 313669-88-4 |
Catalog # | 23269-1 |
Price | $49.00 |
Order / More Info | BMS 986122 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |