Ensifentrine from CAYMAN CHEMICAL COMPANY

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Product NameEnsifentrine
DescriptionA PDE3 inhibitor (IC50 = 0.4 nM); selective for PDE3 over PDE4 (IC50 = 1,479 nM); reduces the phytohemagglutinin-induced proliferation of isolated human monocytes; inhibits LPS-induced increases of TNF-α protein levels in isolated human monocytes (IC50 = 520 nM); increases cAMP levels in isolated human neutrophils at 10 µM; inhibits electric field stimulation-induced contractile responses in isolated guinea pig trachea in a concentration-dependent manner; intranasal administration inhibits histamine-induced bronchoconstriction and tracheal edema in guinea pigs at 25% w/w
Size1 mg
Concentrationn/a
Applicationsn/a
Other NamesRPL 554|VMX 554
Gene, Accession, CAS #CAS: 1884461-72-6
Catalog #38761-1
Price$30.00
Order / More InfoEnsifentrine from CAYMAN CHEMICAL COMPANY
Product Specific Referencesn/a
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
CAYMAN CHEMICAL COMPANY
1180 East Ellsworth Road
Ann Arbor MI 48108
P: (734) 971-3335
P: (800) 364-9897 (USA & Canada only)
F: (734) 971-3640

Customer Service: custserv@caymanchem.com
Technical Support: techserv@caymanchem.com
Sales: sales@caymanchem.com

http://www.caymanchem.com

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