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Product Name | Rolapitant |
Description | A potent NK1 receptor antagonist (Ki = 0.66 nM for the human receptor); greater than 1,000-fold selective for NK1 over NK2 and NK3 and lacks activity in a panel of 100 receptors, transporters, enzymes, and ion channels; prevents apomorphine- and cisplatin-induced emesis in ferrets (ED50s = 0.03 and 0.07 mg/kg, respectively) |
Size | 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | varubi SCH-619734SCH619734 NK-1 2 3 GR73632 |
Gene, Accession, CAS # | CAS: 552292-08-7 |
Catalog # | 23906-5 |
Price | $116 |
Order / More Info | Rolapitant from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |