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Product Name | SGC-GAK-1 |
Description | A GAK inhibitor (Ki = 3.1 nM); >50-fold selective for GAK over a panel of 400 kinases at 1 µM but does bind to RIPK2 (IC50 = 360 nM in a BRET engagement assay); reduces the viability of LNCaP and 22Rv1 prostate cancer cells (IC50s = 0.65 and 0.17 µM, respectively); inhibits dengue virus infection in Huh7 cells (EC50 = 0.08 µM) |
Size | 25 mg |
Concentration | n/a |
Applications | n/a |
Other Names | SGC-GAK1 SGCGAK1 SGCGAK-1 RIPK-2 22-Rv1 Huh-7 |
Gene, Accession, CAS # | CAS: 2226517-76-4 |
Catalog # | 33229-25 |
Price | $127.00 |
Order / More Info | SGC-GAK-1 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |