VU0240551 |
A KCC2 inhibitor (IC50 = 568 nM); selectively inhibits KCC2 over NKCC1 (IC… |
5 mg |
29790-5 |
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VU0240551 |
A KCC2 inhibitor (IC50 = 568 nM); selectively inhibits KCC2 over NKCC1 (IC… |
50 mg |
29790-50 |
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VU0255035 |
A selective, competitive orthosteric antagonist of the muscarinic M1 recep… |
10 mg |
19353-10 |
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VU0255035 |
A selective, competitive orthosteric antagonist of the muscarinic M1 recep… |
50 mg |
19353-50 |
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VU0357121 |
A positive allosteric modulator of mGluR5 (EC50 = 33 nM); selective for mG… |
10 mg |
22199-10 |
More Info
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VU0357121 |
A positive allosteric modulator of mGluR5 (EC50 = 33 nM); selective for mG… |
25 mg |
22199-25 |
More Info
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VU0357121 |
A positive allosteric modulator of mGluR5 (EC50 = 33 nM); selective for mG… |
5 mg |
22199-5 |
More Info
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VU0357121 |
A positive allosteric modulator of mGluR5 (EC50 = 33 nM); selective for mG… |
50 mg |
22199-50 |
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VU0359595 |
A highly selective inhibitor of PLD1 (IC50 = 3.7 nM) versus PLD2 (IC50 = 6… |
1 mg |
10955-1 |
More Info
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VU0359595 |
A highly selective inhibitor of PLD1 (IC50 = 3.7 nM) versus PLD2 (IC50 = 6… |
10 mg |
10955-10 |
More Info
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VU0359595 |
A highly selective inhibitor of PLD1 (IC50 = 3.7 nM) versus PLD2 (IC50 = 6… |
25 mg |
10955-25 |
More Info
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VU0359595 |
A highly selective inhibitor of PLD1 (IC50 = 3.7 nM) versus PLD2 (IC50 = 6… |
5 mg |
10955-5 |
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VU0360223 |
A selective, negative allosteric modulator of the mGlu5 (IC50 = 61 nM; Ki… |
1 mg |
11995-1 |
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VU0360223 |
A selective, negative allosteric modulator of the mGlu5 (IC50 = 61 nM; Ki… |
10 mg |
11995-10 |
More Info
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VU0360223 |
A selective, negative allosteric modulator of the mGlu5 (IC50 = 61 nM; Ki… |
5 mg |
11995-5 |
More Info
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VU0360223 |
A selective, negative allosteric modulator of the mGlu5 (IC50 = 61 nM; Ki… |
50 mg |
11995-50 |
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VU0361737 |
A selective PAM of mGluR4, displaying EC50 values of 110 and 240 nM for ra… |
1 mg |
16295-1 |
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VU0361737 |
A selective PAM of mGluR4, displaying EC50 values of 110 and 240 nM for ra… |
10 mg |
16295-10 |
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VU0361737 |
A selective PAM of mGluR4, displaying EC50 values of 110 and 240 nM for ra… |
5 mg |
16295-5 |
More Info
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VU0364439 |
A positive allosteric modulator of mGluR4; potentiates glutamate responses… |
1 mg |
16296-1 |
More Info
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VU0364439 |
A positive allosteric modulator of mGluR4; potentiates glutamate responses… |
10 mg |
16296-10 |
More Info
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VU0364439 |
A positive allosteric modulator of mGluR4; potentiates glutamate responses… |
5 mg |
16296-5 |
More Info
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VU0364439 |
A positive allosteric modulator of mGluR4; potentiates glutamate responses… |
50 mg |
16296-50 |
More Info
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VU0364770 |
A positive allosteric modulator of metabotropic glutamate receptor 4 (mGlu… |
10 mg |
22927-10 |
More Info
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VU0364770 |
A positive allosteric modulator of metabotropic glutamate receptor 4 (mGlu… |
25 mg |
22927-25 |
More Info
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VU0364770 |
A positive allosteric modulator of metabotropic glutamate receptor 4 (mGlu… |
5 mg |
22927-5 |
More Info
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VU0364770 |
A positive allosteric modulator of metabotropic glutamate receptor 4 (mGlu… |
50 mg |
22927-50 |
More Info
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VU0365114 |
A positive allosteric modulator of muscarinic M5 receptors; increases ACh-… |
10 mg |
33709-10 |
More Info
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VU0365114 |
A positive allosteric modulator of muscarinic M5 receptors; increases ACh-… |
100 mg |
33709-100 |
More Info
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VU0365114 |
A positive allosteric modulator of muscarinic M5 receptors; increases ACh-… |
50 mg |
33709-50 |
More Info
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VU0409551 |
An mGluR5 PAM; induces calcium mobilization in HEK293 cells expressing hum… |
1 mg |
18042-1 |
More Info
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VU0409551 |
An mGluR5 PAM; induces calcium mobilization in HEK293 cells expressing hum… |
10 mg |
18042-10 |
More Info
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VU0409551 |
An mGluR5 PAM; induces calcium mobilization in HEK293 cells expressing hum… |
25 mg |
18042-25 |
More Info
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VU0409551 |
An mGluR5 PAM; induces calcium mobilization in HEK293 cells expressing hum… |
5 mg |
18042-5 |
More Info
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VU0467154 |
A positive allosteric modulator of the M4 muscarinic acetylcholine recepto… |
1 mg |
25555-1 |
More Info
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VU0467154 |
A positive allosteric modulator of the M4 muscarinic acetylcholine recepto… |
10 mg |
25555-10 |
More Info
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VU0467154 |
A positive allosteric modulator of the M4 muscarinic acetylcholine recepto… |
25 mg |
25555-25 |
More Info
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VU0467154 |
A positive allosteric modulator of the M4 muscarinic acetylcholine recepto… |
5 mg |
25555-5 |
More Info
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VU0483605 |
A selective mGluR1 PAM (EC50s = 0.39 and 0.36 µM for human and rat r… |
1 mg |
16941-1 |
More Info
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VU0483605 |
A selective mGluR1 PAM (EC50s = 0.39 and 0.36 µM for human and rat r… |
10 mg |
16941-10 |
More Info
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VU0483605 |
A selective mGluR1 PAM (EC50s = 0.39 and 0.36 µM for human and rat r… |
5 mg |
16941-5 |
More Info
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VU0661013 |
An Mcl-1 inhibitor (Ki = 97 pM); selective for Mcl-1 over Bcl-xL and Bcl-2… |
1 mg |
39524-1 |
More Info
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VU0661013 |
An Mcl-1 inhibitor (Ki = 97 pM); selective for Mcl-1 over Bcl-xL and Bcl-2… |
10 mg |
39524-10 |
More Info
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VU0661013 |
An Mcl-1 inhibitor (Ki = 97 pM); selective for Mcl-1 over Bcl-xL and Bcl-2… |
5 mg |
39524-5 |
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VUF 10166 |
A 5-HT3A antagonist (Ki = 0.04 nM); selective for 5-HT3A over 5-HT3AB rece… |
10 mg |
31423-10 |
More Info
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VUF 10166 |
A 5-HT3A antagonist (Ki = 0.04 nM); selective for 5-HT3A over 5-HT3AB rece… |
100 mg |
31423-100 |
More Info
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VUF 10166 |
A 5-HT3A antagonist (Ki = 0.04 nM); selective for 5-HT3A over 5-HT3AB rece… |
25 mg |
31423-25 |
More Info
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VUF 10166 |
A 5-HT3A antagonist (Ki = 0.04 nM); selective for 5-HT3A over 5-HT3AB rece… |
50 mg |
31423-50 |
More Info
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VUF 5574 |
An adenosine A3 receptor antagonist (Ki = 4.03 nM for the recombinant huma… |
1 mg |
27676-1 |
More Info
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VUF 5574 |
An adenosine A3 receptor antagonist (Ki = 4.03 nM for the recombinant huma… |
10 mg |
27676-10 |
More Info
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VUF 5574 |
An adenosine A3 receptor antagonist (Ki = 4.03 nM for the recombinant huma… |
5 mg |
27676-5 |
More Info
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VUF10460 |
A histamine H4 receptor agonist (Kis = 5.01 and 14.13 for the human and ra… |
1 mg |
14665-1 |
More Info
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VUF10460 |
A histamine H4 receptor agonist (Kis = 5.01 and 14.13 for the human and ra… |
10 mg |
14665-10 |
More Info
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VUF10460 |
A histamine H4 receptor agonist (Kis = 5.01 and 14.13 for the human and ra… |
25 mg |
14665-25 |
More Info
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VUF10460 |
A histamine H4 receptor agonist (Kis = 5.01 and 14.13 for the human and ra… |
5 mg |
14665-5 |
More Info
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VUF8430 (hydrobromide) |
A histamine H4 receptor agonist (Ki = 31.6 nM); selective for histamine H4… |
1 mg |
27682-1 |
More Info
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VUF8430 (hydrobromide) |
A histamine H4 receptor agonist (Ki = 31.6 nM); selective for histamine H4… |
10 mg |
27682-10 |
More Info
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VUF8430 (hydrobromide) |
A histamine H4 receptor agonist (Ki = 31.6 nM); selective for histamine H4… |
25 mg |
27682-25 |
More Info
|
VUF8430 (hydrobromide) |
A histamine H4 receptor agonist (Ki = 31.6 nM); selective for histamine H4… |
5 mg |
27682-5 |
More Info
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VUF 11207 (trifluoroacetate salt) |
A potent CXCR7 receptor agonist (EC50 = 1.6 nM for β-arrestin recruit… |
1 mg |
19812-1 |
More Info
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VUF 11207 (trifluoroacetate salt) |
A potent CXCR7 receptor agonist (EC50 = 1.6 nM for β-arrestin recruit… |
10 mg |
19812-10 |
More Info
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VUF 11207 (trifluoroacetate salt) |
A potent CXCR7 receptor agonist (EC50 = 1.6 nM for β-arrestin recruit… |
5 mg |
19812-5 |
More Info
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VU0134992 (hydrochloride) |
An inhibitor of Kir4.1 (IC50 = 5.2 µM in a thallium flux assay); sel… |
10 mg |
37299-10 |
More Info
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VU0134992 (hydrochloride) |
An inhibitor of Kir4.1 (IC50 = 5.2 µM in a thallium flux assay); sel… |
25 mg |
37299-25 |
More Info
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VU0134992 (hydrochloride) |
An inhibitor of Kir4.1 (IC50 = 5.2 µM in a thallium flux assay); sel… |
5 mg |
37299-5 |
More Info
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VU0134992 (hydrochloride) |
An inhibitor of Kir4.1 (IC50 = 5.2 µM in a thallium flux assay); sel… |
50 mg |
37299-50 |
More Info
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VU0357017 (hydrochloride) |
A selective agonist of M1 mAChRs (Ki = 9.91 µM); selective for M1 ov… |
1 mg |
11939-1 |
More Info
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VU0357017 (hydrochloride) |
A selective agonist of M1 mAChRs (Ki = 9.91 µM); selective for M1 ov… |
10 mg |
11939-10 |
More Info
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VU0357017 (hydrochloride) |
A selective agonist of M1 mAChRs (Ki = 9.91 µM); selective for M1 ov… |
25 mg |
11939-25 |
More Info
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VU0357017 (hydrochloride) |
A selective agonist of M1 mAChRs (Ki = 9.91 µM); selective for M1 ov… |
5 mg |
11939-5 |
More Info
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VU0360172 (hydrochloride) |
A positive allosteric modulator of mGluR5 (Ki = 195 nM); selective for mGl… |
10 mg |
22074-10 |
More Info
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VU0360172 (hydrochloride) |
A positive allosteric modulator of mGluR5 (Ki = 195 nM); selective for mGl… |
25 mg |
22074-25 |
More Info
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VU0360172 (hydrochloride) |
A positive allosteric modulator of mGluR5 (Ki = 195 nM); selective for mGl… |
5 mg |
22074-5 |
More Info
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VU0360172 (hydrochloride) |
A positive allosteric modulator of mGluR5 (Ki = 195 nM); selective for mGl… |
50 mg |
22074-50 |
More Info
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VU0469650 (hydrochloride) |
A negative allosteric mGluR1 modulator; inhibits glutamate-induced calcium… |
1 mg |
32933-1 |
More Info
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