GSK8612 |
A TBK1 inhibitor (IC50 = 158 nM); selective for TBK1 over a panel of 285 k… |
5 mg |
28813-5 |
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GSK8612 |
A TBK1 inhibitor (IC50 = 158 nM); selective for TBK1 over a panel of 285 k… |
50 mg |
28813-50 |
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GSK864 |
An inhibitor of mutant IDH1 (IC50s = 9, 15, and 17 nM for IDH1 mutants R13… |
1 mg |
18762-1 |
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GSK864 |
An inhibitor of mutant IDH1 (IC50s = 9, 15, and 17 nM for IDH1 mutants R13… |
10 mg |
18762-10 |
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GSK864 |
An inhibitor of mutant IDH1 (IC50s = 9, 15, and 17 nM for IDH1 mutants R13… |
5 mg |
18762-5 |
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GSK864 |
An inhibitor of mutant IDH1 (IC50s = 9, 15, and 17 nM for IDH1 mutants R13… |
500 µg |
18762-500 |
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GSK872 |
A selective inhibitor of RIPK3; >1,000-fold selectivity over 300 kinases i… |
1 mg |
23300-1 |
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GSK872 |
A selective inhibitor of RIPK3; >1,000-fold selectivity over 300 kinases i… |
10 mg |
23300-10 |
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GSK872 |
A selective inhibitor of RIPK3; >1,000-fold selectivity over 300 kinases i… |
5 mg |
23300-5 |
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GSK923295 |
A potent inhibitor of CENP-E (Ki = 3.2 nM); causes mitotic cell cycle dela… |
1 mg |
18389-1 |
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GSK923295 |
A potent inhibitor of CENP-E (Ki = 3.2 nM); causes mitotic cell cycle dela… |
10 mg |
18389-10 |
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GSK923295 |
A potent inhibitor of CENP-E (Ki = 3.2 nM); causes mitotic cell cycle dela… |
5 mg |
18389-5 |
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GSK923295 |
A potent inhibitor of CENP-E (Ki = 3.2 nM); causes mitotic cell cycle dela… |
50 mg |
18389-50 |
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GSK963 |
A RIPK1 inhibitor; selective for RIPK1 with 50s = 1 and 4 nM, respectively… |
10 mg |
39900-10 |
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GSK963 |
A RIPK1 inhibitor; selective for RIPK1 with 50s = 1 and 4 nM, respectively… |
25 mg |
39900-25 |
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GSK963 |
A RIPK1 inhibitor; selective for RIPK1 with 50s = 1 and 4 nM, respectively… |
5 mg |
39900-5 |
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GSK963 |
A RIPK1 inhibitor; selective for RIPK1 with 50s = 1 and 4 nM, respectively… |
50 mg |
39900-50 |
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GSK843 |
A RIPK3 inhibitor (IC50 = 6.5 nM); selective for RIPK3 over a panel of 300… |
1 mg |
39835-1 |
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GSK843 |
A RIPK3 inhibitor (IC50 = 6.5 nM); selective for RIPK3 over a panel of 300… |
10 mg |
39835-10 |
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GSK843 |
A RIPK3 inhibitor (IC50 = 6.5 nM); selective for RIPK3 over a panel of 300… |
25 mg |
39835-25 |
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GSK843 |
A RIPK3 inhibitor (IC50 = 6.5 nM); selective for RIPK3 over a panel of 300… |
5 mg |
39835-5 |
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GSK329 |
A TNNI3K inhibitor and sorafenib derivative (IC50 = 10 nM); selective for… |
1 mg |
40666-1 |
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GSK329 |
A TNNI3K inhibitor and sorafenib derivative (IC50 = 10 nM); selective for… |
10 mg |
40666-10 |
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GSK329 |
A TNNI3K inhibitor and sorafenib derivative (IC50 = 10 nM); selective for… |
5 mg |
40666-5 |
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GSK620 |
A BET BD2 inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD… |
10 mg |
36139-10 |
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GSK620 |
A BET BD2 inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD… |
25 mg |
36139-25 |
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GSK620 |
A BET BD2 inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD… |
5 mg |
36139-5 |
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GSK620 |
A BET BD2 inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD… |
50 mg |
36139-50 |
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GSK 417651A |
A TRPC3 and TRPC6 inhibitor (IC50 = ~0.4 µM for both); inhibits migr… |
1 mg |
15268-1 |
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GSK 417651A |
A TRPC3 and TRPC6 inhibitor (IC50 = ~0.4 µM for both); inhibits migr… |
10 mg |
15268-10 |
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GSK 417651A |
A TRPC3 and TRPC6 inhibitor (IC50 = ~0.4 µM for both); inhibits migr… |
25 mg |
15268-25 |
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GSK 417651A |
A TRPC3 and TRPC6 inhibitor (IC50 = ~0.4 µM for both); inhibits migr… |
5 mg |
15268-5 |
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GSK1016790A |
A TRPV4 agonist that has been reported to elicit calcium influx in HEK cel… |
1 mg |
17289-1 |
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GSK1016790A |
A TRPV4 agonist that has been reported to elicit calcium influx in HEK cel… |
10 mg |
17289-10 |
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GSK1016790A |
A TRPV4 agonist that has been reported to elicit calcium influx in HEK cel… |
25 mg |
17289-25 |
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GSK1016790A |
A TRPV4 agonist that has been reported to elicit calcium influx in HEK cel… |
5 mg |
17289-5 |
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GSK137647A |
A selective agonist of GPR120 (EC50s = 0.5, 0.63, and 0.79 µM for hu… |
10 mg |
17712-10 |
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GSK137647A |
A selective agonist of GPR120 (EC50s = 0.5, 0.63, and 0.79 µM for hu… |
25 mg |
17712-25 |
More Info
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GSK137647A |
A selective agonist of GPR120 (EC50s = 0.5, 0.63, and 0.79 µM for hu… |
5 mg |
17712-5 |
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GSK137647A |
A selective agonist of GPR120 (EC50s = 0.5, 0.63, and 0.79 µM for hu… |
50 mg |
17712-50 |
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GSK1702934A |
A TRPC3 and TRPC6 activator; induces TRPC3- and TRPC6-dependent currents i… |
1 mg |
34576-1 |
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GSK1702934A |
A TRPC3 and TRPC6 activator; induces TRPC3- and TRPC6-dependent currents i… |
10 mg |
34576-10 |
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GSK1702934A |
A TRPC3 and TRPC6 activator; induces TRPC3- and TRPC6-dependent currents i… |
5 mg |
34576-5 |
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GSK180736A |
A ROCK1 and GRK2 inhibitor (IC50s = 14 and 0.77 µM, respectively); s… |
10 mg |
26182-10 |
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GSK180736A |
A ROCK1 and GRK2 inhibitor (IC50s = 14 and 0.77 µM, respectively); s… |
25 mg |
26182-25 |
More Info
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GSK180736A |
A ROCK1 and GRK2 inhibitor (IC50s = 14 and 0.77 µM, respectively); s… |
5 mg |
26182-5 |
More Info
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GSK180736A |
A ROCK1 and GRK2 inhibitor (IC50s = 14 and 0.77 µM, respectively); s… |
50 mg |
26182-50 |
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GSK1838705A |
An IGF-1R and IR inhibitor (IC50s = 2 and 1.6 nM, respectively); selective… |
10 mg |
24904-10 |
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GSK1838705A |
An IGF-1R and IR inhibitor (IC50s = 2 and 1.6 nM, respectively); selective… |
25 mg |
24904-25 |
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GSK1838705A |
An IGF-1R and IR inhibitor (IC50s = 2 and 1.6 nM, respectively); selective… |
5 mg |
24904-5 |
More Info
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