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Product Name | Dilazep (hydrochloride) |
Description | An ENT1 inhibitor (IC50 = 17.5 nM); selective for ENT1 over ENT2 (IC50 = 8,800 nM); increases adenosine-induced relaxation of isolated guinea pig taenia caeci strips at 0.03 and 0.3 µM; decreases calcium-induced contractions in isolated guinea pig taenia caeci strips at 1, 5, and 10 µM; reduces heart rate and systolic, mean, and diastolic aortic pressure and increases left ventricular blood flow in anesthetized dogs at 0.2 mg/kg, i.v.; reduces aortic platelet adhesion and aggregation in a rabbit model of aortic injury-induced thrombosis at 0.1 mg/kg |
Size | 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 126748-76-3 35898-87-4 ENT 1 2 comelian cormelian |
Gene, Accession, CAS # | CAS: 20153-98-4 |
Catalog # | 29761-5 |
Price | $62.00 |
Order / More Info | Dilazep (hydrochloride) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |