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Product Name | VER-246608 |
Description | A pan-PDHK inhibitor (IC50s = 35, 84, 40, and 91 nM for PDHK1, -2, -3, and -4, respectively); selective for PDHKs over Hsp90 (IC50 = >100 µM), as well as a panel of 97 kinases at 10 µM; decreases L-lactate production in PC3 cells cultured in D-glucose- and L-glutamine-depleted media at 10 and 20 µM; reduces the growth of, and induces cell cycle arrest at the G1 phase in, serum-starved PC3 cells at 20 µM |
Size | 25 mg |
Concentration | n/a |
Applications | n/a |
Other Names | VER246608 PDHK2 PDHK3 PDHK4 Hsp-90 |
Gene, Accession, CAS # | CAS: 1684386-71-7 |
Catalog # | 19182-25 |
Price | $448.00 |
Order / More Info | VER-246608 from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |