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Product Name | CPI-203 |
Description | Purity >98%. CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM (BRD4 α-screen assay). MW: 399.9 |
Size | 5 mg, 10 mg, 25 mg |
Concentration | 0.1 mM: 25.01 mL (1 mg); 125.03 mL (5 mg); 250.06mL (10 mg). 0.5 mM: 5 mL (1 mg); 25.01 mL (5 mg); 50.01 mL (10 mg). 1 mM: 2.5 mL (1 mg); 12.5 mL (5 mg); 25.01 mL (10 mg). 5 mM: 0.5 mL (1 mg); 2.5 mL (5 mg); 5 mL (10 mg) |
Applications | n/a |
Other Names | n/a |
Gene, Accession, CAS # | CAS: 1446144-04-2 |
Catalog # | MBS385350 |
Price | $150, $230, $420 |
Order / More Info | CPI-203 from MYBIOSOURCE INC. |
Product Specific References | Derenzini E,.et al. BET Inhibition-Induced GSK3 Feedback Enhances Lymphoma Vulnerability to PI3K Inhibitors, Cell Rep, 2018, Aug 21;24(8):2155-2166 PMID: 30134175 |