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Product Name | Azamulin |
Description | Purity ≥98% by HPLC. Azamulin is a derivative of the antibiotic pleuromutilin. It is a highly selective inhibitor of the CYP3A family (IC50 = 0.03-0.24 muM as reported in Stresser et al.; DMD; January 2004 vol. 32 no. 1 p105-112). Azamulin is a 15 and 13 fold more potent inhibitor of CYP3A4 compared to CYP3A5 or CYP3A7 respectively making it very useful for CYP3A4 activity assays and can be used as a benchmark in CYP3A4 inhibitor screening assays. It is at least 100 fold selective over other CYP isoforms (except CYP2J2 ~ 50-fold). MW: 478.65 |
Size | 1 mg, 5 mg |
Concentration | n/a |
Applications | n/a |
Other Names | n/a |
Gene, Accession, CAS # | CAS: 76530-44-4 |
Catalog # | MBS845469 |
Price | $125, $305 |
Order / More Info | Azamulin from MYBIOSOURCE INC. |
Product Specific References | n/a |