A-769662 |
A direct activator of AMPK (EC50 = 116 nM in a cell-free assay); allosteri… |
5 mg |
11900-5 |
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A-769662 |
A direct activator of AMPK (EC50 = 116 nM in a cell-free assay); allosteri… |
50 mg |
11900-50 |
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A-770041 |
An orally bioavailable LCK kinase inhibitor (IC50 = 0.147 µM); selec… |
1 mg |
32854-1 |
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A-770041 |
An orally bioavailable LCK kinase inhibitor (IC50 = 0.147 µM); selec… |
5 mg |
32854-5 |
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A-77-01 |
A potent inhibitor of the TGF-β1 receptor ALK5 (IC550 = 25 nM), block… |
1 mg |
18396-1 |
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A-77-01 |
A potent inhibitor of the TGF-β1 receptor ALK5 (IC550 = 25 nM), block… |
10 mg |
18396-10 |
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A-77-01 |
A potent inhibitor of the TGF-β1 receptor ALK5 (IC550 = 25 nM), block… |
25 mg |
18396-25 |
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A-77-01 |
A potent inhibitor of the TGF-β1 receptor ALK5 (IC550 = 25 nM), block… |
5 mg |
18396-5 |
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A-771726 |
An active metabolite of leflunomide; inhibits DHODH (IC50 = 0.23 µM)… |
10 mg |
14404-10 |
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A-771726 |
An active metabolite of leflunomide; inhibits DHODH (IC50 = 0.23 µM)… |
25 mg |
14404-25 |
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A-771726 |
An active metabolite of leflunomide; inhibits DHODH (IC50 = 0.23 µM)… |
5 mg |
14404-5 |
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A-784168 |
A TRPV1 competitive antagonist; inhibits capsaicin-induced activation of T… |
1 mg |
32855-1 |
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A-784168 |
A TRPV1 competitive antagonist; inhibits capsaicin-induced activation of T… |
10 mg |
32855-10 |
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A-784168 |
A TRPV1 competitive antagonist; inhibits capsaicin-induced activation of T… |
25 mg |
32855-25 |
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A-784168 |
A TRPV1 competitive antagonist; inhibits capsaicin-induced activation of T… |
5 mg |
32855-5 |
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A-796260 |
A synthetic CB that shows high selectivity for the CB2 receptor (Ki = 0.77… |
1 mg |
11606-1 |
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A-796260 |
A synthetic CB that shows high selectivity for the CB2 receptor (Ki = 0.77… |
10 mg |
11606-10 |
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A-796260 |
A synthetic CB that shows high selectivity for the CB2 receptor (Ki = 0.77… |
5 mg |
11606-5 |
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A-803467 |
A sodium channel blocker with high-affinity and selectivity for inhibiting… |
10 mg |
10012588-10 |
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A-803467 |
A sodium channel blocker with high-affinity and selectivity for inhibiting… |
100 mg |
10012588-100 |
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A-803467 |
A sodium channel blocker with high-affinity and selectivity for inhibiting… |
5 mg |
10012588-5 |
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A-803467 |
A sodium channel blocker with high-affinity and selectivity for inhibiting… |
50 mg |
10012588-50 |
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A-804598 |
A potent and selective competitive antagonist of the P2X7 receptor (IC50s… |
10 mg |
20060-10 |
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A-804598 |
A potent and selective competitive antagonist of the P2X7 receptor (IC50s… |
25 mg |
20060-25 |
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A-804598 |
A potent and selective competitive antagonist of the P2X7 receptor (IC50s… |
5 mg |
20060-5 |
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A-804598 |
A potent and selective competitive antagonist of the P2X7 receptor (IC50s… |
50 mg |
20060-50 |
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A-834735 |
An indole-derived CB that acts as a full agonist at both the CB1 and CB2 r… |
1 mg |
11163-1 |
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A-834735 |
An indole-derived CB that acts as a full agonist at both the CB1 and CB2 r… |
10 mg |
11163-10 |
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A-834735 |
An indole-derived CB that acts as a full agonist at both the CB1 and CB2 r… |
5 mg |
11163-5 |
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A-836339 |
A synthetic CB which has a higher affinity for the peripheral CB2 receptor… |
1 mg |
13898-1 |
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A-836339 |
A synthetic CB which has a higher affinity for the peripheral CB2 receptor… |
10 mg |
13898-10 |
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A-836339 |
A synthetic CB which has a higher affinity for the peripheral CB2 receptor… |
5 mg |
13898-5 |
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A-839977 |
A P2X7 receptor antagonist; inhibits BzATP-evoked intracellular calcium in… |
1 mg |
30934-1 |
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A-839977 |
A P2X7 receptor antagonist; inhibits BzATP-evoked intracellular calcium in… |
10 mg |
30934-10 |
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A-839977 |
A P2X7 receptor antagonist; inhibits BzATP-evoked intracellular calcium in… |
5 mg |
30934-5 |
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A-841720 |
A noncompetitive antagonist of mGluR1 (IC50 = 10.7 nM); selective over mGl… |
1 mg |
21807-1 |
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A-841720 |
A noncompetitive antagonist of mGluR1 (IC50 = 10.7 nM); selective over mGl… |
10 mg |
21807-10 |
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A-841720 |
A noncompetitive antagonist of mGluR1 (IC50 = 10.7 nM); selective over mGl… |
5 mg |
21807-5 |
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A-867744 |
A positive allosteric modulator of α7 nAChRs; selective for α7… |
10 mg |
32974-10 |
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A-867744 |
A positive allosteric modulator of α7 nAChRs; selective for α7… |
100 mg |
32974-100 |
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A-867744 |
A positive allosteric modulator of α7 nAChRs; selective for α7… |
50 mg |
32974-50 |
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A-922500 |
A potent inhibitor of DGAT-1 (IC50s = 7 and 24 nM, for human and mouse, re… |
1 mg |
10012708-1 |
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A-922500 |
A potent inhibitor of DGAT-1 (IC50s = 7 and 24 nM, for human and mouse, re… |
10 mg |
10012708-10 |
More Info
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A-922500 |
A potent inhibitor of DGAT-1 (IC50s = 7 and 24 nM, for human and mouse, re… |
25 mg |
10012708-25 |
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A-922500 |
A potent inhibitor of DGAT-1 (IC50s = 7 and 24 nM, for human and mouse, re… |
5 mg |
10012708-5 |
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A-939572 |
A stearoyl-CoA desaturase 1 inhibitor (IC50 = 6.3 nM) that induces cell de… |
10 mg |
19123-10 |
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A-939572 |
A stearoyl-CoA desaturase 1 inhibitor (IC50 = 6.3 nM) that induces cell de… |
5 mg |
19123-5 |
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A-939572 |
A stearoyl-CoA desaturase 1 inhibitor (IC50 = 6.3 nM) that induces cell de… |
50 mg |
19123-50 |
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A-966492 |
A dual inhibitor of PARP1 and PARP2 (Kis = 1 and 1.5 nM, respectively); re… |
1 mg |
26378-1 |
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A-966492 |
A dual inhibitor of PARP1 and PARP2 (Kis = 1 and 1.5 nM, respectively); re… |
10 mg |
26378-10 |
More Info
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