Edit |   |
---|---|
Product Name | Darusentan |
Description | Darusentan is a selective antagonist of ET-A Endothelin receptors, inhibiting Endothelin-1 radioligand binding to ET-A and ET-B receptors with Ki of 6 nM and 371 nM, respectively1. in vitro Darusentan inhibits Endothelin-induced vascular contractility in isolated endothelium-denuded rat aortic rings with pA2 of 8.12. Darusentan is orally bioavailable and active in vivo3. Synthetic. Purity >99%. MW: 410.43 |
Size | 10 mg |
Concentration | 1 nM - 1 µM. |
Applications | n/a |
Other Names | n/a |
Gene, Accession, CAS # | CAS: 171714-84-4 |
Catalog # | D-265 |
Price | please inquire |
Order / More Info | Darusentan from ALOMONE LABS |
Product Specific References | n/a |
U.S.A. OFFICE
Toll free phone: 1800-618-1644 / 1800-791-3904
Toll free fax: 1888-454-7276 / 1800-791-3912