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Product Name | BQ-123 trifluoroacetate |
Description | BQ-123, a cyclic peptide, is a potent and selective antagonist of ET-A endothelin receptors, exhibiting a 1000-fold selectivity for ET-A over ET-B receptors (inhibiting endothelin-1 radioligand binding to ET-A and ET-B with IC50 of 22 nM and 18 µM, respectively). In vitro, BQ-123 inhibits endothelin-1 induced contractions of porcine coronary artery with KB of 40 nM1. Synthetic. Purity >98%. MW: 724.74 |
Size | 10 mg |
Concentration | 10 nM - 10 µM. |
Applications | n/a |
Other Names | n/a |
Gene, Accession, CAS # | CAS: 136553-81-6 |
Catalog # | B-186 |
Price | please inquire |
Order / More Info | BQ-123 trifluoroacetate from ALOMONE LABS |
Product Specific References | n/a |
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