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Product Name | Clemastine (fumarate) |
Description | A histamine H1 receptor antagonist (Ki = 0.26 nM); selective for the histamine H1 receptor over mAChRs (Ki = 16 nM), as well as over σ1 and σ2 and α2A-, α2B-, and α2C-adrenergic receptors (Kis = 67, 15, 1,365, 691, and 545 nM, respectively); reduces ovalbumin-induced bronchial obstruction in ovalbumin-sensitized guinea pigs alone or in combination with cimetidine at 0.12 mg/kg; decreases SARS-CoV-2 replication in SARS-CoV-2-infected Vero E6 cells (EC50 = 0.95 µM) |
Size | 1 g |
Concentration | n/a |
Applications | n/a |
Other Names | 52205-67-1 15686-51-8 meclastin antihistamines anti-histamines anti histamines H1 receptors antagonists muscarinic P2X7 bronchoconstriction asthma airways hyperresponsiveness allosteric signaling inhibits inhibitors inhibitions agasten aloginan alphamin anhistan bravegly hydrogen fuluminol HS 592 HS592 HS-592 unbestan kinotomin lacretin lecasol maikohis mallermin F mallermin-F marsthine masletine meclastine mecloprodine piloral reconin tavegil tavegyl tavist telgin telgin-G Gs trabest xolamin neurosciences inflammation allergy asthma purinoceptor genes |
Gene, Accession, CAS # | CAS: 14976-57-9 |
Catalog # | 14637-1 |
Price | $410.00 |
Order / More Info | Clemastine (fumarate) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |