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Product Name | CP 100,356 (hydrochloride) |
Description | A P-glycoprotein inhibitor (IC50 = 0.5 µM); selective for P-gp over MRP2 at 15 µM, CYP1A2, CYP2C9, CYP2C19, CYP2D6, and CYP3A4 (IC50s = >50 µM for all), and OATP2B1 (IC50 = ~66 µM) but does inhibit BCRP (IC50 = 1.5 µM); increases the rate of prazosin clearance in rats at 24 mg/kg when administered in combination with prazosin |
Size | 1 mg |
Concentration | n/a |
Applications | n/a |
Other Names | 142716-85-6 Pglycoprotein CP100356 Pgp CYP450 CYP 1A2 2C9 2C19 2D6 3A4 OAT P1B1 |
Gene, Accession, CAS # | CAS: 142715-48-8 |
Catalog # | 32853-1 |
Price | $62.00 |
Order / More Info | CP 100,356 (hydrochloride) from CAYMAN CHEMICAL COMPANY |
Product Specific References | n/a |