GSK189254 |
A histamine H3 receptor antagonist (Kis = 0.13, 0.68, and 1.74 nM for the… |
5 mg |
36705-5 |
More Info
|
GSK1940029 |
A stearoyl-CoA desaturase inhibitor; increases palmitate-induced phosphory… |
1 mg |
36704-1 |
More Info
|
GSK1940029 |
A stearoyl-CoA desaturase inhibitor; increases palmitate-induced phosphory… |
10 mg |
36704-10 |
More Info
|
GSK1940029 |
A stearoyl-CoA desaturase inhibitor; increases palmitate-induced phosphory… |
25 mg |
36704-25 |
More Info
|
GSK1940029 |
A stearoyl-CoA desaturase inhibitor; increases palmitate-induced phosphory… |
5 mg |
36704-5 |
More Info
|
GSK2018682 |
An S1P1 and S1P5 receptor agonist; selective for S1P1 and S1P5 over S1P2,… |
10 mg |
31437-10 |
More Info
|
GSK2018682 |
An S1P1 and S1P5 receptor agonist; selective for S1P1 and S1P5 over S1P2,… |
25 mg |
31437-25 |
More Info
|
GSK2018682 |
An S1P1 and S1P5 receptor agonist; selective for S1P1 and S1P5 over S1P2,… |
5 mg |
31437-5 |
More Info
|
GSK2018682 |
An S1P1 and S1P5 receptor agonist; selective for S1P1 and S1P5 over S1P2,… |
50 mg |
31437-50 |
More Info
|
GSK2033 |
An antagonist of LXRα and LXRβ (IC50s = 0.1 and 0.398 µM,… |
1 mg |
25443-1 |
More Info
|
GSK2033 |
An antagonist of LXRα and LXRβ (IC50s = 0.1 and 0.398 µM,… |
10 mg |
25443-10 |
More Info
|
GSK2033 |
An antagonist of LXRα and LXRβ (IC50s = 0.1 and 0.398 µM,… |
5 mg |
25443-5 |
More Info
|
GSK2126458 |
A potent inhibitor of PI3K isoforms (Kis = 19, 130, 24, and 60 pM for p110… |
1 mg |
17377-1 |
More Info
|
GSK2126458 |
A potent inhibitor of PI3K isoforms (Kis = 19, 130, 24, and 60 pM for p110… |
10 mg |
17377-10 |
More Info
|
GSK2126458 |
A potent inhibitor of PI3K isoforms (Kis = 19, 130, 24, and 60 pM for p110… |
5 mg |
17377-5 |
More Info
|
GSK2126458 |
A potent inhibitor of PI3K isoforms (Kis = 19, 130, 24, and 60 pM for p110… |
50 mg |
17377-50 |
More Info
|
GSK2190915 |
A selective inhibitor of human FLAP (IC50 = 2.9 nM); selective for FLAP ov… |
1 mg |
28600-1 |
More Info
|
GSK2193874 |
A potent, selective antagonist of TRPV4 channels, blocking the influx of c… |
1 mg |
17715-1 |
More Info
|
GSK2193874 |
A potent, selective antagonist of TRPV4 channels, blocking the influx of c… |
10 mg |
17715-10 |
More Info
|
GSK2193874 |
A potent, selective antagonist of TRPV4 channels, blocking the influx of c… |
25 mg |
17715-25 |
More Info
|
GSK2193874 |
A potent, selective antagonist of TRPV4 channels, blocking the influx of c… |
5 mg |
17715-5 |
More Info
|
GSK2194069 |
An inhibitor of fatty acid synthase (IC50 = 7.7 nM in an assay detecting r… |
1 mg |
20022-1 |
More Info
|
GSK2194069 |
An inhibitor of fatty acid synthase (IC50 = 7.7 nM in an assay detecting r… |
5 mg |
20022-5 |
More Info
|
GSK2194069 |
An inhibitor of fatty acid synthase (IC50 = 7.7 nM in an assay detecting r… |
500 µg |
20022-500 |
More Info
|
GSK2245035 |
A TLR7 agonist; selectively induces the production of IFN-α over TNF… |
1 mg |
33171-1 |
More Info
|
GSK2245035 |
A TLR7 agonist; selectively induces the production of IFN-α over TNF… |
10 mg |
33171-10 |
More Info
|
GSK2245035 |
A TLR7 agonist; selectively induces the production of IFN-α over TNF… |
5 mg |
33171-5 |
More Info
|
GSK2256098 |
A FAK inhibitor; selective for FAK over 261 kinases; inhibits FAK autophos… |
1 mg |
22955-1 |
More Info
|
GSK2256098 |
A FAK inhibitor; selective for FAK over 261 kinases; inhibits FAK autophos… |
10 mg |
22955-10 |
More Info
|
GSK2256098 |
A FAK inhibitor; selective for FAK over 261 kinases; inhibits FAK autophos… |
25 mg |
22955-25 |
More Info
|
GSK2256098 |
A FAK inhibitor; selective for FAK over 261 kinases; inhibits FAK autophos… |
5 mg |
22955-5 |
More Info
|
GSK2269557 |
A selective PI3Kδ inhibitor (pKi = 9.9) that is active in a brown No… |
1 mg |
17388-1 |
More Info
|
GSK2269557 |
A selective PI3Kδ inhibitor (pKi = 9.9) that is active in a brown No… |
10 mg |
17388-10 |
More Info
|
GSK2269557 |
A selective PI3Kδ inhibitor (pKi = 9.9) that is active in a brown No… |
25 mg |
17388-25 |
More Info
|
GSK2269557 |
A selective PI3Kδ inhibitor (pKi = 9.9) that is active in a brown No… |
5 mg |
17388-5 |
More Info
|
GSK2292767 |
A potent and selective inhibitor of PI3Kδ (Ki = 79 pM); has >1,000-f… |
1 mg |
21757-1 |
More Info
|
GSK2292767 |
A potent and selective inhibitor of PI3Kδ (Ki = 79 pM); has >1,000-f… |
10 mg |
21757-10 |
More Info
|
GSK2292767 |
A potent and selective inhibitor of PI3Kδ (Ki = 79 pM); has >1,000-f… |
25 mg |
21757-25 |
More Info
|
GSK2292767 |
A potent and selective inhibitor of PI3Kδ (Ki = 79 pM); has >1,000-f… |
5 mg |
21757-5 |
More Info
|
GSK2330672 |
An ASBT inhibitor (IC50s = 42, 2.1, and 1.9 nM for human, mouse, and rat A… |
1 mg |
23843-1 |
More Info
|
GSK2330672 |
An ASBT inhibitor (IC50s = 42, 2.1, and 1.9 nM for human, mouse, and rat A… |
10 mg |
23843-10 |
More Info
|
GSK2330672 |
An ASBT inhibitor (IC50s = 42, 2.1, and 1.9 nM for human, mouse, and rat A… |
5 mg |
23843-5 |
More Info
|
GSK2334470 |
A selective PDK1 inhibitor (IC50 = ~10 nM) that even at 100-fold higher co… |
10 mg |
18095-10 |
More Info
|
GSK2334470 |
A selective PDK1 inhibitor (IC50 = ~10 nM) that even at 100-fold higher co… |
25 mg |
18095-25 |
More Info
|
GSK2334470 |
A selective PDK1 inhibitor (IC50 = ~10 nM) that even at 100-fold higher co… |
5 mg |
18095-5 |
More Info
|
GSK2334470 |
A selective PDK1 inhibitor (IC50 = ~10 nM) that even at 100-fold higher co… |
50 mg |
18095-50 |
More Info
|
GSK25 |
A ROCK1 inhibitor (IC50 = 7 nM for the human kinase); selective over RSK1… |
1 mg |
39163-1 |
More Info
|
GSK25 |
A ROCK1 inhibitor (IC50 = 7 nM for the human kinase); selective over RSK1… |
10 mg |
39163-10 |
More Info
|
GSK25 |
A ROCK1 inhibitor (IC50 = 7 nM for the human kinase); selective over RSK1… |
5 mg |
39163-5 |
More Info
|
GSK25 |
A ROCK1 inhibitor (IC50 = 7 nM for the human kinase); selective over RSK1… |
500 µg |
39163-500 |
More Info
|